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Expired Canadian patentCanada

Tetrahydro-naphthalene derivatives as vanilloid receptor antagonists

CA 2508845 C · Owner: Tsukimi, Yasuhiro · Inventors: Mogi, Muneto; Shiroo, Masahiro; Kokubo, Toshio

CIPO record

Overview

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Its claims, description and drawings are in the Canadian Patents Database.

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Abstract From the Canadian patent

This invention relates to tetrahydro-naphthalene derivatives and salts thereof which is useful as an active ingredient of pharmaceutical preparations. The tetrahydro-naphthalene derivatives of the present invention have an excellent activity as VR1 antagonist and useful for the prophylaxis and treatment of diseases associated with VR1 activity, in particular for the treatment of urinary incontinence, urge urinary incontinence overactive bladder, chronic , pain, neuropathic pain postoperative pain, rheumatoid arthritic pain neuralgia, neuropathies, algesia, nerve injury ischaemia, neurodegeneration, stroke, inflammatory disorders asthma and COPD.

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Listed from its CIPO record in Patent Yard's archive of Canadian patents past their term. Its claims, description and drawings are in the CIPO record and on Google Patents, and the Claude kit works from them.

Why it's free to use

  • Filed November 28, 2003 and granted February 21, 2012. A Canadian patent filed from October 1, 1989 lasts 20 years from filing, so its term ended November 28, 2023.
  • A certificate of supplementary protection adds at most two years for a drug, so even that would have ended by November 28, 2025.
  • We check Canadian rights only. A patent in its family in another country could still be in force: check its family on Google Patents.
FiledNovember 28, 2003
GrantedFebruary 21, 2012
Term endedNovember 28, 2023
Patent numberCA 2508845 C
Classification (IPC)C07C275/32 +2 more

Timeline

Timeline From CIPO dates

2004200620082010201220142016201820202022Application filedNov 28, 2003Patent grantedFeb 21, 2012Term endedNov 28, 2023

Sources & verification

Everything on this page comes from the CIPO record linked above. Contains information licensed under the Open Government Licence – Canada.