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Expired Canadian patentCanada

7-amino-2-heptenoates and their use in the preparation of methylphenidate

CA 2243544 C · Owner: Fox, Martin Edward · Inventors: Fox, Martin Edward; Paul, Jane Marie

CIPO record

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Its claims, description and drawings are in the Canadian Patents Database.

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Abstract From the Canadian patent

Novel compounds are of the formula Y1Y2N-(CH2)4-CH=C(Ph)-X wherein Y1 and Y2 are independently H or a removable blocking group or Y1 and Y2 together are a , removable divalent blocking group; and X is COOCH3 or a group convertible thereto. Such a compound may be cyclised by Michael addition, to give , methylphenidate if necessary after removing blocking group(s) and converting X to COOCH3.

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Listed from its CIPO record in Patent Yard's archive of Canadian patents past their term. Its claims, description and drawings are in the CIPO record and on Google Patents, and the Claude kit works from them.

Why it's free to use

  • Filed March 21, 1997 and granted November 19, 2002. A Canadian patent filed from October 1, 1989 lasts 20 years from filing, so its term ended March 21, 2017.
  • A certificate of supplementary protection adds at most two years for a drug, so even that would have ended by March 21, 2019.
  • We check Canadian rights only. A patent in its family in another country could still be in force: check its family on Google Patents.
FiledMarch 21, 1997
GrantedNovember 19, 2002
Term endedMarch 21, 2017
Patent numberCA 2243544 C
Classification (IPC)C07D211/34 +2 more

Timeline

Timeline From CIPO dates

1998200020022004200620082010201220142016Application filedMarch 21, 1997Patent grantedNov 19, 2002Term endedMarch 21, 2017

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Everything on this page comes from the CIPO record linked above. Contains information licensed under the Open Government Licence – Canada.