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Expired Canadian patentCanada

Indole derivatives

CA 2178161 C · Owner: Pfizer Inc. · Inventors: Wythes, Martin James; Macor, John Eugene

CIPO record

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Abstract From the Canadian patent

Compounds of the formula , I wherein n is 0 1, or 2; X is chlorine, bromine, or iodine; R1 is hydrogen; R2 is selected from hydrogen halogen, cyano, -OR4 -(CH2)m-(C=O)NR5R6 -(CH2)m-SO2NR5R6, -(CH2)m-NR7(C=O)R8 --(CH2)m-NR7SO2R8 -(CH2) m-S(O)xR8, -(CH2)m-NR,(C=O)NR5R6 -(CH2)m-NR,(C=O)OR9, and -CH=CH(CH2)yR10; R3 is C1 to C6 linear or branched alkyl and the pharmaceutically acceptable salts thereof are new. These compounds are useful psychotherapeutics and are potent serotonin (5-HT1) agonists and may be used in the treatment of depression anxiety, eating disorders, obesity, drug abuse cluster headache, migraine, pain, chronic paroxysmal hemicrania and headache associated with vascular …

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Listed from its CIPO record in Patent Yard's archive of Canadian patents past their term. Its claims, description and drawings are in the CIPO record and on Google Patents, and the Claude kit works from them.

Why it's free to use

  • Filed June 4, 1996 and granted December 18, 2001. A Canadian patent filed from October 1, 1989 lasts 20 years from filing, so its term ended June 4, 2016.
  • A certificate of supplementary protection adds at most two years for a drug, so even that would have ended by June 4, 2018.
  • We check Canadian rights only. A patent in its family in another country could still be in force: check its family on Google Patents.
FiledJune 4, 1996
GrantedDecember 18, 2001
Term endedJune 4, 2016
Patent numberCA 2178161 C
Classification (IPC)C07D403/06 +2 more

Timeline

Timeline From CIPO dates

1997199920012003200520072009201120132015Application filedJune 4, 1996Patent grantedDec 18, 2001Term endedJune 4, 2016

Sources & verification

Everything on this page comes from the CIPO record linked above. Contains information licensed under the Open Government Licence – Canada.