6-oxoazepinoindole compounds, processes and intermediates for their preparation and pharmaceutical compositions containing them

Abstract From the Canadian patent

Pharmacologically active compounds corresponding to the general formula I, I, in which, R1 represents hydrogen a lower alkyl or cycloalkyl-, alkyl group or an optionally substituted phenyllower alkyl group, R2 denotes hydrogen or a lower alkyl group optionally substituted in the .alpha.-position to the nitrogen atom by lower alkoxy, R3 denotes hydrogen, lower alkyl lower alkoxy, halogen, or hydroxyl, n represents 1 or if the -(CH2)n- chain is in the 4-, position of the ring structure also represents 2, R4 denotes hydrogen lower alkyl, cycloalkyl, cyclo-, alkyl-lower alkyl or an optionally substituted phenyl-lower alkyl group, and, R5 denotes hydrogen lower alkyl, cycloalkyl, cyclo-, …