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Expired Canadian patentCanada

Bis-(1h-indol-3-yl)-maleinimide derivatives and their use as pharmaceuticals

CA 2015996 C · Owner: Barth, Hubert · Inventors: Barth, Hubert; Betche, Hans-Jurgen; Schachtele, Christoph

CIPO record

Overview

Drawings and full text

Its claims, description and drawings are in the Canadian Patents Database.

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Abstract From the Canadian patent

The present invention provides bis-(1H-indol-3-yl)maleinimide derivatives and the pharmacologically acceptable salts thereof, processes for the preparation of these compounds and pharmaceutical compositions containing them for the treatment of heart and blood vessel diseases such as, thromboses, arteriosclerosis, hypertension of inflammatory processes, allergies, cancer and certain degenerative damages of the central nervous system, as well as of diseases of the immune system and viral diseases. The maleinimide derivatives of the invention are of formula I, and an example is the compound in which R1 is methyl and R2 R4, R5, R8 and R9 are each hydrogen.

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Listed from its CIPO record in Patent Yard's archive of Canadian patents past their term. Its claims, description and drawings are in the CIPO record and on Google Patents, and the Claude kit works from them.

Why it's free to use

  • Filed May 3, 1990 and granted August 28, 2001. A Canadian patent filed from October 1, 1989 lasts 20 years from filing, so its term ended May 3, 2010.
  • A certificate of supplementary protection adds at most two years for a drug, so even that would have ended by May 3, 2012.
  • We check Canadian rights only. A patent in its family in another country could still be in force: check its family on Google Patents.
FiledMay 3, 1990
GrantedAugust 28, 2001
Term endedMay 3, 2010
Patent numberCA 2015996 C
Classification (IPC)C07D401/14 +2 more

Timeline

Timeline From CIPO dates

1991199319951997199920012003200520072009Application filedMay 3, 1990Patent grantedAug 28, 2001Term endedMay 3, 2010

Sources & verification

Everything on this page comes from the CIPO record linked above. Contains information licensed under the Open Government Licence – Canada.