Spermicidal vaginal composition comprising 1,2-benzisothiazole derivatives

Abstract From the Canadian patent

SPERMICIDAL VAGINAL COMPOSITIONS COMPRISING 1,2-BENZISOTHIAZOLE DERIVATIVES", Abstract Or the disclosure A spermicidal vaginal composition comprises a spermicidal-effective amount of a 1,2-benzisothiazole derivative having the general formula (I), wherein: X is either O or S;, y is H; NO2; an halogen atom or an alkyl radical having from 1 to 4 carbon atoms; and, R is H; a straight or branched alkyl or alkenyl radical having from 1 to 6 carbon atoms, optionally substituted by one or more hydroxyl, tertiary amino and alkoxyl groups; a cycloaliphatic radical having from 3 to 8 carbon atoms; an alkyl radical optionally substituted by halogen atoms alkyl or alkoxyl radicals; an aralkyl radical …